2 uger), blev der i kliniske forsøg givet en initialdosis på 100 mg i 3 dage for at opnå hurtig steady- state koncentrationer af A771726.
Due to the very long half-life of A771726 (approximately 2 weeks), a loading dose of 100 mg for 3 days was used in clinical studies to facilitate the rapid attainment of steady-state levels of A771726.