Valsartan udskilles primært ved galdeudskillelse i fæces (cirka 83% af dosis) og renalt i urin (cirka 13% af dosis), hovedsageligt som uomdannet stof.
Valsartan is primarily eliminated by biliary excretion in faeces (about 83% of dose) and renally in urine (about 13% of dose), mainly as unchanged drug.