hat
Tcheke gout, mibolerone non chimik, CAS No.3704-9-4, te orijinèlman pwodwi kòm yon èd nan kenbe chen fi soti nan ale nan chalè. Teknikman li konsidere ak Androjen, sepandan, mibolerone tou se trè pwogestasyonèl ki se mekanis a pou efè li yo nan chen fi.An reyalite, mibolerone gen sou de fwa afinite a pou reseptè a pwojestewòn kòm pwojestewòn tèt li. Dwòg sa a te gen yon repitasyon tankou yo te yon trè ki pisan esteroyid itil nan rive mas ak pou agrandisman byen wo ogmante agresyon. Dwòg sa a se dériver ni-19 nan bolasterone epi kòm nandrolone se pi plis ki pi pisan ak plis progestational pase testostewòn, se konsa se ka a ak mibolerone konpare ak bolasterone. Anplis de sa nan gwoup la methyl nan C-7 pa sèlman ogmante AR ak PR aktivite, men tou ogmante toksisite la nan molekil la. Mibolerone se yon derive nan nortestosterone (nandrolone); sepandan, li pa metabolize nan yon metabolit dihydronandrolone mwens ki pisan akòz efè a pwoteje nan gwoup la methyl 7-alfa.
eng
Cheque drops, chemical name mibolerone,CAS No.3704-9-4, was originally produced as an aid in keeping female dogs from going into heat. Technically it is considered and androgen, however, mibolerone is also very progestational which is the mechanism for its effects in female dogs.In fact, mibolerone has about twice the affinity for the progesterone receptor as progesterone itself. This drug had a reputation as being a very potent steroid useful in attaining mass and for drastically increasing aggression. This drug is the nor-19 derivative of bolasterone and as nandrolone is more potent and more progestational than testosterone, so is the case with mibolerone compared to bolasterone. The addition of the methyl group at C-7 not only increases AR and PR activity but also increases the toxicity of the molecule. Mibolerone is a derivative of nortestosterone (nandrolone); however, it is not metabolized to a less potent dihydronandrolone metabolite due to the shielding effect of the 7-alpha methyl group.