List of steroidal antiandrogens
# List of steroidal antiandrogens

This is a list of steroidal antiandrogens.

## Progesterone derivatives

* 11α-Hydroxyprogesterone = 11α-hydroxyprogesterone
* Chlormadinone acetate = $17α-acetoxy-6-chloro-δ^6-progesterone$
* Clometerone (L-38000) = 6α-chloro-16α-methylprogesterone
* Cyproterone (SH-80881) = $1,2α-methylene-6-chloro-δ^6-17α-hydroxyprogesterone$
* Cyproterone acetate = $1,2α-methylene-6-chloro-δ^6-17α-acetoxyprogesterone$
* Edogestrone (PH-218) = 17α-acetoxy-3,3-ethylenedioxy-6-methylpregn-5-en-20-one
* Medrogestone = $6,17α-dimethyl-δ^6-progesterone$
* Megestrol acetate = $17α-acetoxy-δ^6-6-methylprogesterone$
* Nomegestrol acetate = $17α-acetoxy-δ^6-6-methyl-19-norprogesterone$
* Osaterone acetate (TZP-4238) = $17α-acetoxy-6-chloro-2-oxa-δ^6-progesterone$

## Testosterone derivatives

* Abiraterone (CB-7598) = 17-(3-pyridinyl)androsta-5,16-dien-3β-ol
* Abiraterone acetate = 17-(3-pyridinyl)androsta-5,16-dien-3β-ol acetate
* Benorterone (SKF-7690, FC-612) = 17α-methyl-B-nortestosterone
* BOMT (Ro 7-2340) = 6α-bromo-4-oxa-17α-methyl-4,5α-dihydrotestosterone
* Delanterone (GBR-21162) = $17β-dehydroxy-1α-methyl-δ^{16}-testosterone$
* Dienogest = $17α-cyanomethyl-19-nor-δ^{9(10)}-testosterone$
* Epitestosterone = 17α-epitestosterone
* Galeterone (TOK-001, VN/124-1) = 17-(1H-benzimidazol-1-yl)androsta-5,16-dien-3β-ol
* Metogest (SC-14207) = 16,16-dimethyl-19-nortestosterone
* Mifepristone = $11β-[p-(dimethylamino)phenyl]-17-(1-propynyl)-δ^9-19-nortestosterone$
* Oxendolone (TSAA-291) = 16β-ethyl-19-nortestosterone
* Rosterolone (SH-434, 17α-propylmesterolone) = 1α-methyl-17α-propyl-4,5α-dihydrotestosterone
* Topterone (WIN-17665) = 17α-propyltestosterone
* Trimethyltrienolone (R-2956, RU-2956) = $2α,2β,17α-trimethyl-19-nor-δ^{9,11}-testosterone$
* Zanoterone (WIN-49596) = (5α,17α)-1'-(methylsulfonyl)-1'-H-pregn-20-yno[3,2-c]pyrazol-17-ol

## Spirolactone derivatives

* SC-5233 (spirolactone) = 17α-(2-carboxyethyl)testosterone γ-lactone
* SC-8109 = 19-norspirolactone
* Canrenone (aldadiene) = $Δ^6-spirolactone$
* Dicirenone (SC-26304) = 7α-carboxyisopropylspirolactone
* Drospirenone = 6β,7β:15β,16β-dimethylenespirolactone
* Mespirenone (ZK-94679) = $Δ^1-7α-acetylthio-15β,16β-methylenespirolactone$
* Mexrenone (ZK-32055, SC-25152) = 7α-(methoxycarbonyl)spirolactone
* Prorenone (SC-23133) = 6α,7α-methylenespirolactone
* Spironolactone = 7α-acetylthiospirolactone
* Spirorenone (ZK-35973) = $Δ^1-6β,7β:15β,16β-dimethylenespirolactone$
* Spiroxasone = 7α-acetylthiospirolactone with the ketone group removed from the C17α spirolactone ring

## Cortisol derivatives

* 9,11-Dehydrocortexolone 17α-butyrate (CB-03-04) = 17α-(butyryloxy)-9,11-didehydrodeoxycorticosterone
* Clascoterone (CB-03-01; cortexolone 17α-propionate, 11-deoxycortisol 17α-propionate) = 17α-(propionyloxy)deoxycorticosterone

## Others

* Guggulsterone = pregna-4,17-diene-3,16-dione
* Nordinone = 11α-hydroxy-17,17-dimethyl-18-norandrosta-4,13-dien-3-one
