A-372159
# A-372159

A-372159 is a drug which acts as a potent and selective partial agonist for the $5HT_{2C}$ receptor, with more than 100x selectivity over the closely related $5-HT_{2B}$ receptor and a Ki of 3nM. It has been found to produce anorectic effects in animal studies and produced significant weight loss in rats with no development of tolerance or serious side effects.

